Pirenzepine 2HCl

Active Pharmaceutical Ingredients 2025-03-03

Catalog ID80018938

CAS NO.29868-97-1

Purity 99%

MDL NumberMFCD00055214

EINEC249-907-5

Molecular formula C19H21N5O2.2HCl

Molecular weight 424.3242

Category Details
Chemical Properties Molecular formula: C19H23Cl2N5O2<br> Molecular weight: 460.78
Physical Properties Appearance: White crystalline powder<br> Melting point: 240–243°C
Mechanism of Action Selective muscarinic receptor antagonist, primarily targeting M1 receptors in the gastric mucosa. Reduces gastric acid and pepsin secretion by blocking these receptors.
Therapeutic Uses Used for treating peptic ulcers, gastric ulcers, and duodenal ulcers. Also used for acute gastric mucosal bleeding and conditions with excessive gastric acid secretion.
Storage Conditions Store in a cool, dry place, protected from light and moisture.
Safety Information Acute toxicity LD50 in mice: 3000 mg/kg (oral), 109 mg/kg (intravenous).
Synonyms Pirenzepine dihydrochloride, Gastrozepin, LS 519

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