Pilsicainide hydrochloride CAS NO.88069-49-2
Active Pharmaceutical Ingredients 2025-03-03
Catalog ID80017072
CAS NO.88069-49-2
Purity 98+%
MDL NumberMFCD00903769
EINEC Molecular Formula C17H24N2O.HCl
Molecular Weight 308.8462
| Aspect | Details |
|---|---|
| Chemical Structure | – Molecular Formula: C₁₇H₂₅ClN₂O<br>- Molecular Weight: 308.8 g/mol |
| Mechanism of Action | Pilsicainide hydrochloride is a class IC antiarrhythmic agent. It works by blocking fast sodium channels in cardiac cells, thereby reducing the rate of depolarization and slowing the conduction of electrical impulses in the heart. |
| Clinical Uses | – Used for the treatment of supraventricular and ventricular arrhythmias.<br>- Also indicated for the management of atrial fibrillation. |
| Pharmacokinetics | – Absorption: Rapidly absorbed after oral or intravenous administration.<br>- Distribution: Widely distributed in body tissues.<br>- Metabolism: Metabolized in the liver.<br>- Excretion: Primarily excreted in urine. |
| Physical Properties | – Appearance: White to off-white powder.<br>- Solubility: Soluble in water. |
| Storage Conditions | Store in a cool, dry place, protected from moisture and light. |
| Side Effects | Common side effects include nausea, dizziness, and headache. Serious side effects may include prolonged QT interval and torsades de pointes. |
| Regulatory Status | Approved for use in the treatment of arrhythmias in several countries |
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